A convenient methodology for the synthesis of functionalized nitrogen mustards

A.V.Reddy, J.Gopalakrishna, Ke

Abstract

A short protocol for the synthesis of functionalized bis(chloroethyl)amines (nitrogen mustards) has been described via the nucleophilic substitution of allylic bromides derived fromBaylis-Hillman alcoholswith diethanolamine followed by dichlorination.

Relevant Publications in Organic Chemistry : An Indian Journal